IMIDAZOLE DERIVATIVES AS PRODRUGS OF DICLOFENAC

Claus Selch Larsen; Susan Weng Larsen; Mette Agergaard Thing; Jesper Langgaard Kristensen; HENRIK JENSEN,; JESPER ØSTERGAARD,

IMIDAZOLE DERIVATIVES AS PRODRUGS OF DICLOFENAC

Claus Selch Larsen (Opfinder), Susan Weng Larsen (Opfinder), Mette Agergaard Thing (Opfinder), Jesper Langgaard Kristensen (Opfinder), HENRIK JENSEN, (Opfinder), JESPER ØSTERGAARD, (Opfinder)

Publikation: Patent

Abstract

The present invention relates to a compound of formula (I): wherein R1is R3-IPU and R2 is the acyloxy residue of diclofenac, and specified by the following structures: (II), (III) wherein OH-R3-IPU is selected from (IV) and R4 and R5 may be the same or different selected from H and CH3 and salts, solvates and hydrates thereof. The compounds are used for the treatment of pain such as postoperative pain following arthroscopic surgery.

Originalsprog	Engelsk
IPC	A61P 29/ 00 A I
Patentnummer	WO2016066612
Land/Område	Danmark
Prioritetsdato	28/10/2014
Prioritetsnummer	DK20140070657
Status	Udgivet - 6 maj 2016

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Citationsformater

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title = "IMIDAZOLE DERIVATIVES AS PRODRUGS OF DICLOFENAC",

abstract = "The present invention relates to a compound of formula (I): wherein R1is R3-IPU and R2 is the acyloxy residue of diclofenac, and specified by the following structures: (II), (III) wherein OH-R3-IPU is selected from (IV) and R4 and R5 may be the same or different selected from H and CH3 and salts, solvates and hydrates thereof. The compounds are used for the treatment of pain such as postoperative pain following arthroscopic surgery.",

author = "Larsen, {Claus Selch} and Larsen, {Susan Weng} and Thing, {Mette Agergaard} and Kristensen, {Jesper Langgaard} and HENRIK JENSEN, and JESPER {\O}STERGAARD,",

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day = "6",

language = "English",

type = "Patent",

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TY - PAT

T1 - IMIDAZOLE DERIVATIVES AS PRODRUGS OF DICLOFENAC

AU - Larsen, Claus Selch

AU - Larsen, Susan Weng

AU - Thing, Mette Agergaard

AU - Kristensen, Jesper Langgaard

AU - JENSEN,, HENRIK

AU - ØSTERGAARD,, JESPER

PY - 2016/5/6

Y1 - 2016/5/6

N2 - The present invention relates to a compound of formula (I): wherein R1is R3-IPU and R2 is the acyloxy residue of diclofenac, and specified by the following structures: (II), (III) wherein OH-R3-IPU is selected from (IV) and R4 and R5 may be the same or different selected from H and CH3 and salts, solvates and hydrates thereof. The compounds are used for the treatment of pain such as postoperative pain following arthroscopic surgery.

AB - The present invention relates to a compound of formula (I): wherein R1is R3-IPU and R2 is the acyloxy residue of diclofenac, and specified by the following structures: (II), (III) wherein OH-R3-IPU is selected from (IV) and R4 and R5 may be the same or different selected from H and CH3 and salts, solvates and hydrates thereof. The compounds are used for the treatment of pain such as postoperative pain following arthroscopic surgery.

M3 - Patent

M1 - WO2016066612

ER -