New practical access to 2-azatryptophans and dehydro derivatives via the Wittig–Horner reaction

François Crestey; Valerie Collot; Silvia Stiebing; Jean-Francois Lohier; Jana Sopkova-de Oliveira Santos; Sylvain Rault

doi:10.1016/j.tetlet.2007.02.042

New practical access to 2-azatryptophans and dehydro derivatives via the Wittig–Horner reaction

François Crestey, Valerie Collot, Silvia Stiebing, Jean-Francois Lohier, Jana Sopkova-de Oliveira Santos, Sylvain Rault

Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › peer review

14 Citationer (Scopus)

Abstract

The Wittig–Horner reaction of protected 3-formylindazoles 1 with (±)-N-(benzyloxycarbonyl)-α-phosphonoglycine trimethyl ester 2 has been developed as a new practical synthesis of dehydro 2-azatryptophans and amino acid derivatives. The preparation of 5-bromo-3-formylindazole is discussed.

Originalsprog	Engelsk
Tidsskrift	Tetrahedron Letters
Vol/bind	48
Udgave nummer	14
Sider (fra-til)	2457-2460
ISSN	0040-4039
DOI	https://doi.org/10.1016/j.tetlet.2007.02.042
Status	Udgivet - 15 feb. 2007
Udgivet eksternt	Ja

Adgang til dokumentet

10.1016/j.tetlet.2007.02.042

Citationsformater

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abstract = "The Wittig–Horner reaction of protected 3-formylindazoles 1 with (±)-N-(benzyloxycarbonyl)-α-phosphonoglycine trimethyl ester 2 has been developed as a new practical synthesis of dehydro 2-azatryptophans and amino acid derivatives. The preparation of 5-bromo-3-formylindazole is discussed.",

author = "Fran{\c c}ois Crestey and Valerie Collot and Silvia Stiebing and Jean-Francois Lohier and {Sopkova-de Oliveira Santos}, Jana and Sylvain Rault",

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T1 - New practical access to 2-azatryptophans and dehydro derivatives via the Wittig–Horner reaction

AU - Crestey, François

AU - Collot, Valerie

AU - Stiebing, Silvia

AU - Lohier, Jean-Francois

AU - Sopkova-de Oliveira Santos, Jana

AU - Rault, Sylvain

PY - 2007/2/15

Y1 - 2007/2/15

N2 - The Wittig–Horner reaction of protected 3-formylindazoles 1 with (±)-N-(benzyloxycarbonyl)-α-phosphonoglycine trimethyl ester 2 has been developed as a new practical synthesis of dehydro 2-azatryptophans and amino acid derivatives. The preparation of 5-bromo-3-formylindazole is discussed.

AB - The Wittig–Horner reaction of protected 3-formylindazoles 1 with (±)-N-(benzyloxycarbonyl)-α-phosphonoglycine trimethyl ester 2 has been developed as a new practical synthesis of dehydro 2-azatryptophans and amino acid derivatives. The preparation of 5-bromo-3-formylindazole is discussed.

U2 - 10.1016/j.tetlet.2007.02.042

DO - 10.1016/j.tetlet.2007.02.042

M3 - Journal article

SN - 0040-4039

VL - 48

SP - 2457

EP - 2460

JO - Tetrahedron Letters

JF - Tetrahedron Letters

IS - 14

ER -