Anders A. Jensen

Search results

• 2025

  Detailed functional characterization of four nanobodies as positive allosteric modulators of the human calcium-sensing receptor

  Du, W., Rahman, S. N., Barker, E., Bräuner-Osborne, H., Mathiesen, J. M., Ward, D. T. & Jensen, A. A., 2025, In: Biochemical Pharmacology. 231, 12 p., 116619.

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• 2024

  Discovery and Structure-Activity Relationships of 2,5-Dimethoxyphenylpiperidines as Selective Serotonin 5-HT2A Receptor Agonists

  Rørsted, E. M., Jensen, A. A., Smits, G., Frydenvang, K. & Kristensen, J. L., 2024, In: Journal of Medicinal Chemistry. 69, 9, p. 7224–7244

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• Distinct neurodevelopmental and epileptic phenotypes associated with gain- and loss-of-function GABRB2 variants

  Mohammadi, N. A., Ahring, P. K., Yu Liao, V. W., Chua, H. C., Ortiz de la Rosa, S., Johannesen, K. M., Michaeli-Yossef, Y., Vincent-Devulder, A., Meridda, C., Bruel, A. L., Rossi, A., Patel, C., Klepper, J., Bonanni, P., Minghetti, S., Trivisano, M., Specchio, N., Amor, D., Auvin, S., Baer, S. & 12 others, Meyer, P., Milh, M., Salpietro, V., Maroofian, R., Lemke, J. R., Weckhuysen, S., Christophersen, P., Rubboli, G., Chebib, M., Jensen, A. A., Absalom, N. L. & Møller, R. S., 2024, In: EBioMedicine. 106, 20 p., 105236.

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  3 Citations (Scopus)

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• Heterogeneous Origins of Calcium Homeostasis Disorders Arising From 5 Heterozygous Calcium-Sensing Receptor Variants

  Du, W., Boisen, I. M., Rahman, S. N., Poulsen, N. N., Mathiesen, J. M., Jensen, M. B., Bräuner-Osborne, H. & Jensen, A. A., 2024, (E-pub ahead of print) In: The Journal of clinical endocrinology and metabolism. 16 p.

  Research output: Contribution to journal › Journal article › Research › peer-review

• Loss-of-Function Thr347Ala Variant in the G Protein Subunit-α11 Causes Familial Hypocalciuric Hypercalcemia 2 (FHH2)

  Boisen, I. M., Du, W., Juul, A., Bräuner-Osborne, H., Jensen, A. A. & Blomberg Jensen, M., 2024, (E-pub ahead of print) In: The Journal of clinical endocrinology and metabolism.

  Research output: Contribution to journal › Journal article › Research › peer-review

• Structural insights into GABA_A receptor potentiation by Quaalude

  Chojnacka, W., Teng, J., Kim, J. J., Jensen, A. A. & Hibbs, R. E., 2024, In: Nature Communications. 15, 1, 12 p., 5244.

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  1 Citation (Scopus)

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• Understanding paralogous epilepsy-associated GABA_A receptor variants: Clinical implications, mechanisms, and potential pitfalls

  Kan, A. S. H., Kusay, A. S., Mohammadi, N. A., Lin, S. X. N., Liao, V. W. Y., Lesca, G., Souci, S., Milh, M., Christophersen, P., Chebib, M., Møller, R. S., Absalom, N. L., Jensen, A. A. & Ahring, P. K., 2024, In: Proceedings of the National Academy of Sciences of the United States of America. 121, 50, 11 p., e2413011121.

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• 2023

  Discovery of a Novel Class of Benzimidazole-Based Nicotinic Acetylcholine Receptor Modulators: Positive and Negative Modulation Arising from Overlapping Allosteric Sites

  Zhou, L., Dau, V. & Jensen, A. A., 2023, In: Journal of Medicinal Chemistry. 66, 17, p. 12586–12601

  Research output: Contribution to journal › Journal article › Research › peer-review
  1 Citation (Scopus)

• Evolutionary conservation of Zinc-Activated Channel (ZAC) functionality in mammals: a range of mammalian ZACs assemble into cell surface-expressed functional receptors

  Jensen, A. A., 2023, In: Frontiers in Molecular Biosciences. 10, 11 p., 1265429.

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  2 Citations (Scopus)

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• Identification of 5-HT2 Serotonin Receptor Modulators through the Synthesis of a Diverse, Tropane- and Quinuclidine-alkaloid-Inspired Compound Library

  Yao, R., Jensen, A. A., Bryce-Rogers, H. P., Schultz-Knudsen, K., Zhou, L., Hovendal, N. P., Pedersen, H., Kubus, M., Ulven, T. & Laraia, L., 2023, In: Journal of Medicinal Chemistry. 66, 16, p. 11536-11554

  Research output: Contribution to journal › Journal article › Research › peer-review
  5 Citations (Scopus)

• Introducing Conformational Restraints on 25CN-NBOH: A Selective 5-HT_2A Receptor Agonist

  Marcher-Rørsted, E., Nykodemová, J., Harpsøe, K., Jensen, A. A. & Kristensen, J. L., 2023, In: ACS Medicinal Chemistry Letters. 14, 3, p. 319–325

  Research output: Contribution to journal › Journal article › Research › peer-review

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• In Vitro and In Vivo Evaluation of Pellotine: A Hypnotic Lophophora Alkaloid

  Poulie, C. B. M., Chan, C. B., Parka, A., Lettorp, M., Vos, J., Raaschou, A., Pottie, E., Bundgaard, M. S., Sørensen, L. M. E., Cecchi, C. R., Märcher-Rørsted, E., Bach, A., Herth, M. M., Decker, A., Jensen, A. A., Elfving, B., Kretschmann, A. C., Stove, C. P., Kohlmeier, K. A., Cornett, C. & 3 others, Janfelt, C., Kornum, B. R. & Kristensen, J. L., 2023, In: ACS Pharmacology & Translational Science. 6, 10, p. 1492-1507

  Research output: Contribution to journal › Journal article › Research › peer-review

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  2 Citations (Scopus)

• Ligand selectivity hotspots in serotonin GPCRs

  Simon, I. A., Bjørn-Yoshimoto, W. E., Harpsøe, K., Iliadis, S., Svensson, B., Jensen, A. A. & Gloriam, D. E., 2023, In: Trends in Pharmacological Sciences. 44, 12, p. 978-990

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  7 Citations (Scopus)

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• Repeated low doses of psilocybin increase resilience to stress, lower compulsive actions, and strengthen cortical connections to the paraventricular thalamic nucleus in rats

  Kiilerich, K. F., Lorenz, J., Scharff, M. B., Speth, N., Brandt, T. G., Czurylo, J., Xiong, M., Jessen, N. S., Casado-Sainz, A., Shalgunov, V., Kjaerby, C., Satała, G., Bojarski, A. J., Jensen, A. A., Herth, M. M., Cumming, P., Overgaard, A. & Palner, M., 2023, In: Molecular Psychiatry. 28, 9, p. 3829-3841

  Research output: Contribution to journal › Journal article › Research › peer-review
  14 Citations (Scopus)

• Structure–Activity Assessment and In-Depth Analysis of Biased Agonism in a Set of Phenylalkylamine 5-HT2A Receptor Agonists

  Pottie, E., Poulie, C. B. M., Simon, I. A., Harpsøe, K., D’Andrea, L., Komarov, I. V., Gloriam, D. E., Jensen, A. A., Kristensen, J. L. & Stove, C. P., 2023, In: ACS Chemical Neuroscience. 14, 15, p. 2727–2742

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  6 Citations (Scopus)

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• The Concise Guide to PHARMACOLOGY 2023/24: Ion channels

  Alexander, S. P. H., Mathie, A. A., Peters, J. A., Veale, E. L., Striessnig, J., Kelly, E., Armstrong, J. F., Faccenda, E., Harding, S. D., Davies, J. A., Aldrich, R. W., Attali, B., Baggetta, A. M., Becirovic, E., Biel, M., Bill, R. M., Caceres, A. I., Catterall, W. A., Conner, A. C., Davies, P. & 53 others, De Clerq, K., Delling, M., Di Virgilio, F., Falzoni, S., Fenske, S., Fortuny-Gomez, A., Fountain, S., George, C., Goldstein, S. A. N., Grimm, C., Grissmer, S., Ha, K., Hammelmann, V., Hanukoglu, I., Hu, M., Ijzerman, A. P., Jabba, S. V., Jarvis, M., Jensen, A. A., Jordt, S. E., Kaczmarek, L. K., Kellenberger, S., Kennedy, C., King, B., Kitchen, P., Liu, Q., Lynch, J. W., Meades, J., Mehlfeld, V., Nicke, A., Offermanns, S., Perez-Reyes, E., Plant, L. D., Rash, L., Ren, D., Salman, M. M., Sieghart, W., Sivilotti, L. G., Smart, T. G., Snutch, T. P., Tian, J., Trimmer, J. S., Van den Eynde, C., Vriens, J., Wei, A. D., Winn, B. T., Wulff, H., Xu, H., Yang, F., Fang, W., Yue, L., Zhang, X. & Zhu, M., 2023, In: British Journal of Pharmacology. 180 , Suppl 2, p. S145-S222

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  87 Citations (Scopus)

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• 2022

  Discovery of the First Highly Selective Antagonist of the GluK3 Kainate Receptor Subtype

  Chałupnik, P., Vialko, A., Pickering, D. S., Hinkkanen, M., Donbosco, S., Møller, T. C., Jensen, A. A., Nielsen, B., Bay, Y., Kristensen, A. S., Johansen, T. N., Łątka, K., Bajda, M. & Szymańska, E., 2022, In: International Journal of Molecular Sciences. 23, 15, 16 p., 8797.

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  7 Citations (Scopus)

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• Discovery of β-Arrestin-Biased 25CN-NBOH-Derived 5-HT_2A Receptor Agonists

  Poulie, C. B. M., Pottie, E., Simon, I. A., Harpsøe, K., D'Andrea, L., Komarov, I. V., Gloriam, D. E., Jensen, A. A., Stove, C. P. & Kristensen, J. L., 2022, In: Journal of Medicinal Chemistry. 65, 18, p. 12031–12043

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  11 Citations (Scopus)

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• Strychnine and its mono- and dimeric analogues: a pharmaco-chemical perspective

  Zlotos, D. P., Mandour, Y. M. & Jensen, A. A., 2022, In: Natural Product Reports. 39, 10, p. 1910-1937

  Research output: Contribution to journal › Review › Research › peer-review
  7 Citations (Scopus)
• 2021

  25CN-NBOH: A selective agonist for in vitro and in vivo investigations of the serotonin 2A receptor

  Märcher-Rørsted, E., Jensen, A. A. & Kristensen, J. L., 2021, In: ChemMedChem. 16, 21, p. 3263-3270

  Research output: Contribution to journal › Review › Research › peer-review

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• C-2-Linked Dimeric Strychnine Analogues as Bivalent Ligands Targeting Glycine Receptors

  Zlotos, D. P., Abdelmalek, C. M., Botros, L. S., Banoub, M. M., Mandour, Y. M., Breitinger, U., El Nady, A., Breitinger, H-G., Sotriffer, C., Villmann, C., Jensen, A. A. & Holzgrabe, U., 2021, In: Journal of Natural Products. 84, 2, p. 382-394

  Research output: Contribution to journal › Journal article › Research › peer-review
  2 Citations (Scopus)

• Delineation of the functional properties exhibited by the Zinc-Activated Channel (ZAC) and its high-frequency Thr¹²⁸Ala variant (rs2257020) in Xenopus oocytes

  Madjroh, N., Davies, P. A., Smalley, J. L., Kristiansen, U., Söderhielm, P. C. & Jensen, A. A., 2021, In: Pharmacological Research. 169, 18 p., 105653.

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  5 Citations (Scopus)

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• Discovery and functional characterization of N-(thiazol-2-yl)-benzamide analogs as the first class of selective antagonists of the Zinc-Activated Channel (ZAC)

  Madjroh, N., Mellou, E., Davies, P. A., Söderhielm, P. C. & Jensen, A. A., 2021, In: Biochemical Pharmacology. 193, 16 p., 114782.

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  2 Citations (Scopus)

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• Erythrina Alkaloid Analogues as nAChR Antagonists-A Flexible Platform for Leads in Drug Discovery

  Clementson, S., Matheu, S. A., Rørsted, E. M., Pedersen, H., Jensen, A. A., Clausen, R. P., Vital, P., Glibstrup, E., Jessing, M. & Kristensen, J. L., 2021, In: The Journal of Organic Chemistry. 86, 12, p. 8248-8262

  Research output: Contribution to journal › Journal article › Research › peer-review
  1 Citation (Scopus)

• Probing the molecular basis for signal transduction through the Zinc-Activated Channel (ZAC)

  Madjroh, N., Mellou, E., Æbelø, L., Davies, P. A., Söderhielm, P. C. & Jensen, A. A., 2021, In: Biochemical Pharmacology. 193, 18 p., 114781.

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  9 Citations (Scopus)

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• The concise guide to pharmacology 2021/22: Ion channels

  Alexander, S. P., Mathie, A., Peters, J. A., Veale, E. L., Striessnig, J., Kelly, E., Armstrong, J. F., Faccenda, E., Harding, S. D., Pawson, A. J., Southan, C., Davies, J. A., Aldrich, R. W., Attali, B., Baggetta, A. M., Becirovic, E., Biel, M., Bill, R. M., Catterall, W. A., Conner, A. C. & 38 others, Davies, P., Delling, M., Virgilio, F. D., Falzoni, S., Fenske, S., George, C., Goldstein, S. A. N., Grissmer, S., Ha, K., Hammelmann, V., Hanukoglu, I., Jarvis, M., Jensen, A. A., Kaczmarek, L. K., Kellenberger, S., Kennedy, C., King, B., Kitchen, P., Lynch, J. W., Perez-Reyes, E., Plant, L. D., Rash, L., Ren, D., Salman, M. M., Sivilotti, L. G., Smart, T. G., Snutch, T. P., Tian, J., Trimmer, J. S., Van den Eynde, C., Vriens, J., Wei, A. D., Winn, B. T., Wulff, H., Xu, H., Yue, L., Zhang, X. & Zhu, M., 2021, In: British Journal of Pharmacology. 178 , Suppl. 1, p. S157-S245

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  224 Citations (Scopus)

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• 2020

  Characterization of AN317, a novel selective agonist of α6β2-containing nicotinic acetylcholine receptors

  Sandager-Nielsen, K., Ahring, P. K., Klein, J., van Hout, M., Thaneshwaran, S., Santos, A. B. D., Jacobsen, T. A., Amrutkar, D. V., Peters, D., Jensen, A. A., Kohlmeier, K. A., Christophersen, P. & Dyhring, T., 2020, In: Biochemical Pharmacology. 174, 13 p., 113786.

  Research output: Contribution to journal › Journal article › Research › peer-review
  6 Citations (Scopus)

• Characterization of AN6001, the first positive allosteric modulator of α6β2-containing nicotinic acetylcholine receptors

  van Hout, M., Klein, J., Ahring, P. K., Brown, D. T., Thaneshwaran, S., Brito dos Santos, A., Jensen, A. A., Kohlmeier, K. A., Christophersen, P. & Dyhring, T., 2020, In: Biochemical Pharmacology. 174, 113788.

  Research output: Contribution to journal › Journal article › Research › peer-review
  4 Citations (Scopus)

• Comparison of biophysical properties of α1β2 and α3β2 GABAA receptors in whole-cell patch-clamp electrophysiological recordings

  Olander, E. R., Janzen, D., Villmann, C. & Jensen, A. A., 2020, In: P L o S One. 15, 6, 13 p., e0234080.

  Research output: Contribution to journal › Journal article › Research › peer-review

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  3 Citations (Scopus)

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• Dark Classics in Chemical Neuroscience: NBOMes

  Poulie, C. B. M., Jensen, A. A., Halberstadt, A. & Kristensen, J. L., 2020, In: ACS Chemical Neuroscience. p. 3860–3869 10 p.

  Research output: Contribution to journal › Journal article › Research › peer-review
  41 Citations (Scopus)

• Design, Synthesis, and Pharmacological Characterization of Heterobivalent Ligands for the Putative 5-HT_2A/mGlu₂ Receptor Complex

  Poulie, C. B. M., Liu, N., Jensen, A. A. & Bunch, L., 2020, In: Journal of Medicinal Chemistry. 63, 17, p. 9928-9949 22 p.

  Research output: Contribution to journal › Journal article › Research › peer-review
  12 Citations (Scopus)

• From Methaqualone and Beyond: Structure-Activity Relationship of 6-, 7-, and 8-Substituted 2,3-Diphenyl-quinazolin-4(3H)-ones and in Silico Prediction of Putative Binding Modes of Quinazolin-4(3H)-ones as Positive Allosteric Modulators of GABAA Receptors

  Wang, P-F., Jensen, A. A. & Bunch, L., 2020, In: ACS Chemical Neuroscience. 11, 24, p. 4362-4375

  Research output: Contribution to journal › Journal article › Research › peer-review
  10 Citations (Scopus)

• Functional characterization of 5-HT1A and 5-HT1B serotonin receptor signaling through G-protein-activated inwardly rectifying K+ channels in a fluorescence-based membrane potential assay

  Gadgaard, C. & Jensen, A. A., 2020, In: Biochemical Pharmacology. 175, 13 p., 113870.

  Research output: Contribution to journal › Journal article › Research › peer-review
  9 Citations (Scopus)

• Investigation of the 2,5-dimethoxy motif in phenethylamine Serotonin 2A receptor agonists

  Marcher-Rørsted, E., Halberstadt, A. L., Klein, A. K., Chatha, M., Jademyr, S., Jensen, A. A. & Kristensen, J. L., 2020, In: ACS Chemical Neuroscience. 11, p. 1238-1244

  Research output: Contribution to journal › Letter › Research › peer-review
  14 Citations (Scopus)

• Pharmacological Characterization of the Zinc-Activated Channel: A Cys-Loop Receptor Gated by Zn2+, Cu2+ and Protons

  Madjroh, N., Jensen, A. A. & Davies, P. A., 7 Feb 2020, p. 582A-582A.

  Research output: Contribution to conference › Conference abstract for conference › Research

• The selective 5-HT2A receptor agonist 25CN-NBOH: structure-activity relationship, in vivo pharmacology, and in vitro and ex vivo binding characteristics of [3H]25CN-NBOH

  Jensen, A. A., Halberstadt, A. L., Märcher-Rørsted, E., Odland, A. U., Chatha, M., Speth, N., Liebscher, G., Hansen, M., Bräuner-Osborne, H., Palner, M., Andreasen, J. T. & Kristensen, J. L., 2020, In: Biochemical Pharmacology. 177, 16 p., 113979.

  Research output: Contribution to journal › Journal article › Research › peer-review
  21 Citations (Scopus)

• β-Indolyloxy Functionalized Aspartate Analogs as Inhibitors of the Excitatory Amino Acid Transporters (EAATs)

  Liu, N., Jensen, A. A. & Bunch, L., 2020, In: ACS Medicinal Chemistry Letters. 11, 11, p. 2212-2220 9 p.

  Research output: Contribution to journal › Journal article › Research › peer-review

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  1 Citation (Scopus)
• 2019

  11-Aminostrychnine and N-(Strychnine-11-yl)propionamide: Synthesis, Configuration, and Pharmacological Evaluation at Glycine Receptors

  Zlotos, D. P., Mohsen, A. M. Y., Mandour, Y. M., Marzouk, M. A., Breitinger, U., Villmann, C., Breitinger, H-G., Sotriffer, C., Jensen, A. A. & Holzgrabe, U., 6 Aug 2019, In: Journal of Natural Products. 82, p. 2332-2336

  Research output: Contribution to journal › Journal article › Research › peer-review
  4 Citations (Scopus)

• Design and Synthesis of 2,3-trans-Proline Analogs as Ligands for the Ionotropic Glutamate Receptors and the Excitatory Amino Acid Transporters

  Poulie, C. B. M., Alcaide Lopez, A., Krell-Jørgensen, M. P., Larsen, Y., Astier, E., Bjørn-Yoshimoto, W. E., Yi, F., Syrenne, J. T., Storgaard, M., Nielsen, B., Frydenvang, K. A., Jensen, A. A., Hansen, K. B., Pickering, D. S. & Bunch, L., 19 Jun 2019, In: A C S Chemical Neuroscience. 10, 6, p. 2989-3007 19 p.

  Research output: Contribution to journal › Journal article › Research › peer-review

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  4 Citations (Scopus)

• Developing New 4-PIOL and 4-PHP Analogues for Photoinactivation of γ-Aminobutyric Acid Type A Receptors

  Mortensen, M., Krall, J., Kongstad, K. T., Brygger, B. M., Lenzi, O., Francotte, P., Sørensen, T. E., Nielsen, B., Jensen, A. A., Smart, T. G. & Frølund, B., 2019, In: ACS Chemical Neuroscience. 10, 11, p. 4669-4684

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• Discovery of 2-(Imidazo[1,2-b]pyridazin-2-yl)acetic Acid as a New Class of Ligands Selective for the γ-Hydroxybutyric Acid (GHB) High-Affinity Binding Sites

  Krall, J., Bavo, F., Falk-Petersen, C. B., Jensen, C. H., Nielsen, J. O., Tian, Y., Anglani, V., Kongstad, K. T., Piilgaard, L., Nielsen, B., Gloriam, D. E., Kehler, J., Jensen, A. A., Harpsøe, K., Wellendorph, P. & Frølund, B., 14 Mar 2019, In: Journal of Medicinal Chemistry. 62, 5, p. 2798-2813

  Research output: Contribution to journal › Journal article › Research › peer-review
  14 Citations (Scopus)

• Five-membered N-heterocyclic Scaffolds as Novel Amino Bioisosteres at gamma-Aminobutyric Acid (GABA) Type A Receptors and GABA Transporters

  Giraudo, A., Krall, J., Bavo, F., Nielsen, B., Kongstad, K. T., Rolando, B., De Blasio, R., Gloriam, D. E., Löffler, R., Thiesen, L., Harpsøe, K., Frydenvang, K., Boschi, D., Wellendorph, P., Lolli, M. L., Jensen, A. A. & Frølund, B., 27 Jun 2019, In: Journal of Medicinal Chemistry. 62, 12, p. 5797-5809

  Research output: Contribution to journal › Journal article › Research › peer-review
  20 Citations (Scopus)

• Identification and Structure-Activity Relationship Study of Imidazo[1,2-a]pyridine-3-amines as First Selective Inhibitors of Excitatory Amino Acid Transporter Subtype 3 (EAAT3)

  Wu, P., Bjørn-Yoshimoto, W. E., Staudt, M., Jensen, A. A. & Bunch, L., 2019, In: ACS Chemical Neuroscience. 10, p. 4414-4429

  Research output: Contribution to journal › Journal article › Research › peer-review
  10 Citations (Scopus)

• Modulation of thalamo-cortical activity by the NMDA receptor antagonists ketamine and phencyclidine in the awake freely-moving rat

  Amat-Foraster, M., Celada, P., Richter, U., Jensen, A. A., Plath, N., Artigas, F. & Herrik, K. F., 2019, In: Neuropharmacology. 158, 14 p., 107745.

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• THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: Ion channels

  CGTP Collaborators, Dec 2019, In: British Journal of Pharmacology. 176, Suppl 1, p. S142-S228

  Research output: Contribution to journal › Journal article › Research › peer-review
  292 Citations (Scopus)

• Use of the 4-Hydroxy-Triazole Moiety as a Bioisosteric Tool for the Development of Ionotropic Glutamate Receptor Ligands

  Sainas, S., Temperini, P., Farnsworth, J. C., Yi, F., Møllerud, S., Jensen, A. A., Nielsen, B., Kastrup, J. S. J., Hansen, K. B., Boschi, D., Pickering, D. S., Clausen, R. P. & Lolli, M., 2019, In: Journal of Medicinal Chemistry. 62, p. 4467-4482

  Research output: Contribution to journal › Journal article › Research › peer-review

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  20 Citations (Scopus)

• α-Conotoxin VnIB from Conus ventricosus is a potent and selective antagonist of α6β4* nicotinic acetylcholine receptors

  van Hout, M., Valdes, A., Christensen, S. B., Tran, P. T., Watkins, M., Gajewiak, J., Jensen, A. A., Olivera, B. M. & McIntosh, J. M., 2019, In: Neuropharmacology. 157, 107691.

  Research output: Contribution to journal › Journal article › Research › peer-review

  Open Access
  12 Citations (Scopus)
• 2018

  5-HT2C Receptor Structures Reveal the Structural Basis of GPCR Polypharmacology

  Peng, Y., McCorvy, J. D., Harpsøe, K., Lansu, K., Yuan, S., Popov, P., Qu, L., Pu, M., Che, T., Nikolajsen, L. F., Huang, X., Wu, Y., Shen, L., Bjørn-Yoshimoto, W. E., Ding, K., Wacker, D., Han, G. W., Cheng, J., Katritch, V., Jensen, A. A. & 6 others, Hanson, M. A., Zhao, S., Gloriam, D. E., Roth, B. L., Stevens, R. C. & Liu, Z., 2018, In: Cell. 172, 4, p. 719-730 P719-730.E14.

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• Chemoenzymatic synthesis and pharmacological characterization of functionalized aspartate analogues as novel excitatory amino acid transporter inhibitors

  Fu, H., Zhang, J., Tepper, P. G., Bunch, L., Jensen, A. A. & Poelarends, G. J., 13 Sep 2018, In: Journal of Medicinal Chemistry. 61, 17, p. 7741-7753

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• Conformational transitions of the serotonin 5-HT3 receptor

  Polovinkin, L., Hassaine, G., Perot, J., Neumann, E., Jensen, A. A., Lefebvre, S. N., Corringer, P-J., Neyton, J., Chipot, C., Dehez, F., Schoehn, G. & Nury, H., Nov 2018, In: Nature. 563, 7730, p. 275-279 5 p.

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