4-Hydroxy-1,2,3-triazole moiety as bioisostere of the carboxylic acid function: a novel scaffold to probe the orthosteric gamma-aminobutyric acid receptor binding site

Giraudo Alessandro; Jacob Krall; Birgitte Nielsen; Troels Ersted Sørensen; Kenneth Thermann Kongstad; Rolando Barbara; Boschi Donatella; Bente Frølund; Marco L. Lolli

doi:10.1016/j.ejmech.2018.08.094

4-Hydroxy-1,2,3-triazole moiety as bioisostere of the carboxylic acid function: a novel scaffold to probe the orthosteric gamma-aminobutyric acid receptor binding site

Giraudo Alessandro, Jacob Krall, Birgitte Nielsen, Troels Ersted Sørensen, Kenneth Thermann Kongstad, Rolando Barbara, Boschi Donatella, Bente Frølund, Marco L. Lolli

Research output: Contribution to journal › Journal article › Research › peer-review

30 Citations (Scopus)

Original language	English
Journal	European Journal of Medicinal Chemistry
Volume	158
Pages (from-to)	311-321
Number of pages	11
ISSN	0223-5234
DOIs	https://doi.org/10.1016/j.ejmech.2018.08.094
Publication status	Published - 5 Oct 2018

Access to Document

10.1016/j.ejmech.2018.08.094

Cite this

Alessandro, G., Krall, J., Nielsen, B., Sørensen, T. E., Kongstad, K. T., Barbara, R., Donatella, B., Frølund, B., & Lolli, M. L. (2018). 4-Hydroxy-1,2,3-triazole moiety as bioisostere of the carboxylic acid function: a novel scaffold to probe the orthosteric gamma-aminobutyric acid receptor binding site. European Journal of Medicinal Chemistry, 158, 311-321. https://doi.org/10.1016/j.ejmech.2018.08.094

4-Hydroxy-1,2,3-triazole moiety as bioisostere of the carboxylic acid function: a novel scaffold to probe the orthosteric gamma-aminobutyric acid receptor binding site. / Alessandro, Giraudo; Krall, Jacob; Nielsen, Birgitte et al.
In: European Journal of Medicinal Chemistry, Vol. 158, 05.10.2018, p. 311-321.

Research output: Contribution to journal › Journal article › Research › peer-review

Alessandro, G, Krall, J, Nielsen, B, Sørensen, TE, Kongstad, KT, Barbara, R, Donatella, B, Frølund, B & Lolli, ML 2018, '4-Hydroxy-1,2,3-triazole moiety as bioisostere of the carboxylic acid function: a novel scaffold to probe the orthosteric gamma-aminobutyric acid receptor binding site', European Journal of Medicinal Chemistry, vol. 158, pp. 311-321. https://doi.org/10.1016/j.ejmech.2018.08.094

@article{c9e4c580a7164a0394a6517bb5d2f526,

title = "4-Hydroxy-1,2,3-triazole moiety as bioisostere of the carboxylic acid function: a novel scaffold to probe the orthosteric gamma-aminobutyric acid receptor binding site",

author = "Giraudo Alessandro and Jacob Krall and Birgitte Nielsen and S{\o}rensen, {Troels Ersted} and Kongstad, {Kenneth Thermann} and Rolando Barbara and Boschi Donatella and Bente Fr{\o}lund and Lolli, {Marco L.}",

year = "2018",

month = oct,

day = "5",

doi = "10.1016/j.ejmech.2018.08.094",

language = "English",

volume = "158",

pages = "311--321",

journal = "European Journal of Medicinal Chemistry",

issn = "0223-5234",

publisher = "Elsevier Masson",

}

TY - JOUR

T1 - 4-Hydroxy-1,2,3-triazole moiety as bioisostere of the carboxylic acid function: a novel scaffold to probe the orthosteric gamma-aminobutyric acid receptor binding site

AU - Alessandro, Giraudo

AU - Krall, Jacob

AU - Nielsen, Birgitte

AU - Sørensen, Troels Ersted

AU - Kongstad, Kenneth Thermann

AU - Barbara, Rolando

AU - Donatella, Boschi

AU - Frølund, Bente

AU - Lolli, Marco L.

PY - 2018/10/5

Y1 - 2018/10/5

U2 - 10.1016/j.ejmech.2018.08.094

DO - 10.1016/j.ejmech.2018.08.094

M3 - Journal article

C2 - 30223119

SN - 0223-5234

VL - 158

SP - 311

EP - 321

JO - European Journal of Medicinal Chemistry

JF - European Journal of Medicinal Chemistry

ER -