Allosteric modulation of an excitatory amino acid transporter: The subtype-selective inhibitor UCPH-101 exerts sustained inhibition of EAAT1 through an intramonomeric site in the trimerization domain

Bjarke Abrahamsen; Nicole Schneider; Mette Norman Erichsen; Tri Hien Viet Huynh; Christoph Fahlke; Lennart Bunch; Anders A. Jensen

doi:10.1523/JNEUROSCI.3396-12.2013

Allosteric modulation of an excitatory amino acid transporter: The subtype-selective inhibitor UCPH-101 exerts sustained inhibition of EAAT1 through an intramonomeric site in the trimerization domain

Bjarke Abrahamsen, Nicole Schneider, Mette Norman Erichsen, Tri Hien Viet Huynh, Christoph Fahlke, Lennart Bunch, Anders A. Jensen

Medicinal Chemistry Research

Research output: Contribution to journal › Journal article › Research › peer-review

56 Citations (Scopus)

Original language	English
Journal	Journal of Neuroscience
Volume	33
Issue number	3
Pages (from-to)	1068-1087
ISSN	0270-6474
DOIs	https://doi.org/10.1523/JNEUROSCI.3396-12.2013
Publication status	Published - 2013

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Abrahamsen, B., Schneider, N., Erichsen, M. N., Huynh, T. H. V., Fahlke, C., Bunch, L., & Jensen, A. A. (2013). Allosteric modulation of an excitatory amino acid transporter: The subtype-selective inhibitor UCPH-101 exerts sustained inhibition of EAAT1 through an intramonomeric site in the trimerization domain. Journal of Neuroscience, 33(3), 1068-1087. https://doi.org/10.1523/JNEUROSCI.3396-12.2013

Allosteric modulation of an excitatory amino acid transporter: The subtype-selective inhibitor UCPH-101 exerts sustained inhibition of EAAT1 through an intramonomeric site in the trimerization domain. / Abrahamsen, Bjarke; Schneider, Nicole; Erichsen, Mette Norman et al.
In: Journal of Neuroscience, Vol. 33, No. 3, 2013, p. 1068-1087.

Research output: Contribution to journal › Journal article › Research › peer-review

Abrahamsen, B, Schneider, N, Erichsen, MN, Huynh, THV, Fahlke, C, Bunch, L & Jensen, AA 2013, 'Allosteric modulation of an excitatory amino acid transporter: The subtype-selective inhibitor UCPH-101 exerts sustained inhibition of EAAT1 through an intramonomeric site in the trimerization domain', Journal of Neuroscience, vol. 33, no. 3, pp. 1068-1087. https://doi.org/10.1523/JNEUROSCI.3396-12.2013

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