Chemo-enzymatic synthesis of new 2,4-syn-functionalized (S)-glutamate analogues and structure-activity relationship studies at ionotropic glutamate receptors and excitatory amino acid transporters

Z. Assaf; Anja Probst Larsen; Raminta Venskutonyte; Liwei Han; Bjarke Abrahamsen; Birgitte Nielsen; Michael Gajhede; Jette Sandholm Kastrup; Anders A. Jensen; Darryl S Pickering; Karla  Frydenvang; T Gefflaut; Lennart Bunch

doi:10.1021/jm301433m

Chemo-enzymatic synthesis of new 2,4-syn-functionalized (S)-glutamate analogues and structure-activity relationship studies at ionotropic glutamate receptors and excitatory amino acid transporters

Z. Assaf, Anja Probst Larsen, Raminta Venskutonyte, Liwei Han, Bjarke Abrahamsen, Birgitte Nielsen, Michael Gajhede, Jette Sandholm Kastrup, Anders A. Jensen, Darryl S Pickering, Karla Frydenvang, T Gefflaut, Lennart Bunch

Research output: Contribution to journal › Journal article › Research › peer-review

38 Citations (Scopus)

Original language	English
Journal	Journal of Medicinal Chemistry
Volume	56
Issue number	4
Pages (from-to)	1614-1628
ISSN	0022-2623
DOIs	https://doi.org/10.1021/jm301433m
Publication status	Published - 2013

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10.1021/jm301433m

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Assaf, Z., Larsen, A. P., Venskutonyte, R., Han, L., Abrahamsen, B., Nielsen, B., Gajhede, M., Kastrup, J. S., Jensen, A. A., Pickering, D. S., Frydenvang, K., Gefflaut, T., & Bunch, L. (2013). Chemo-enzymatic synthesis of new 2,4-syn-functionalized (S)-glutamate analogues and structure-activity relationship studies at ionotropic glutamate receptors and excitatory amino acid transporters. Journal of Medicinal Chemistry, 56(4), 1614-1628. https://doi.org/10.1021/jm301433m

Chemo-enzymatic synthesis of new 2,4-syn-functionalized (S)-glutamate analogues and structure-activity relationship studies at ionotropic glutamate receptors and excitatory amino acid transporters. / Assaf, Z.; Larsen, Anja Probst; Venskutonyte, Raminta; Han, Liwei; Abrahamsen, Bjarke; Nielsen, Birgitte ; Gajhede, Michael ; Kastrup, Jette Sandholm ; Jensen, Anders A.; Pickering, Darryl S ; Frydenvang, Karla ; Gefflaut, T; Bunch, Lennart.

In: Journal of Medicinal Chemistry, Vol. 56, No. 4, 2013, p. 1614-1628.

Research output: Contribution to journal › Journal article › Research › peer-review

Assaf, Z, Larsen, AP, Venskutonyte, R, Han, L, Abrahamsen, B, Nielsen, B , Gajhede, M , Kastrup, JS , Jensen, AA , Pickering, DS , Frydenvang, K, Gefflaut, T & Bunch, L 2013, 'Chemo-enzymatic synthesis of new 2,4-syn-functionalized (S)-glutamate analogues and structure-activity relationship studies at ionotropic glutamate receptors and excitatory amino acid transporters', Journal of Medicinal Chemistry, vol. 56, no. 4, pp. 1614-1628. https://doi.org/10.1021/jm301433m

Assaf, Z. ; Larsen, Anja Probst ; Venskutonyte, Raminta ; Han, Liwei ; Abrahamsen, Bjarke ; Nielsen, Birgitte ; Gajhede, Michael ; Kastrup, Jette Sandholm ; Jensen, Anders A. ; Pickering, Darryl S ; Frydenvang, Karla ; Gefflaut, T ; Bunch, Lennart. / Chemo-enzymatic synthesis of new 2,4-syn-functionalized (S)-glutamate analogues and structure-activity relationship studies at ionotropic glutamate receptors and excitatory amino acid transporters. In: Journal of Medicinal Chemistry. 2013 ; Vol. 56, No. 4. pp. 1614-1628.

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AU - Venskutonyte, Raminta

AU - Han, Liwei

AU - Abrahamsen, Bjarke

AU - Nielsen, Birgitte

AU - Gajhede, Michael

AU - Kastrup, Jette Sandholm

AU - Jensen, Anders A.

AU - Pickering, Darryl S

AU - Frydenvang, Karla

AU - Gefflaut, T

AU - Bunch, Lennart

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