Chemoenzymatic synthesis and pharmacological characterization of functionalized aspartate analogues as novel excitatory amino acid transporter inhibitors

Haigen Fu; J. Zhang; P.G. Tepper; Lennart Bunch; Anders A. Jensen; G.J. Poelarends

doi:10.1021/acs.jmedchem.8b00700

Chemoenzymatic synthesis and pharmacological characterization of functionalized aspartate analogues as novel excitatory amino acid transporter inhibitors

Haigen Fu, J. Zhang, P.G. Tepper, Lennart Bunch, Anders A. Jensen, G.J. Poelarends

Medicinal Chemistry Research

Research output: Contribution to journal › Journal article › Research › peer-review

18 Citations (Scopus)

228 Downloads (Pure)

Original language	English
Journal	Journal of Medicinal Chemistry
Volume	61
Issue number	17
Pages (from-to)	7741-7753
ISSN	0022-2623
DOIs	https://doi.org/10.1021/acs.jmedchem.8b00700
Publication status	Published - 13 Sep 2018

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Chemoenzymatic synthesis and pharmacological characterization of functionalized aspartate analogues as novel excitatory amino acid transporter inhibitors. / Fu, Haigen; Zhang, J.; Tepper, P.G.; Bunch, Lennart ; Jensen, Anders A.; Poelarends, G.J.

In: Journal of Medicinal Chemistry, Vol. 61, No. 17, 13.09.2018, p. 7741-7753 .

Research output: Contribution to journal › Journal article › Research › peer-review

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AU - Jensen, Anders A.

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