Selective Inhibitors of Glial GABA Uptake: Synthesis, Absolute Stereochemistry, and Pharmacology of the Enantiomers of 3-Hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazole (exo-THPO) and Analogues

Erik Falch; Bente Frølund; null Perregaard; Connie Sanchez; Birgitte Søkilde; Anders Buur; Anette Hansen; Karla Andrea Frydenvang; Lotte Brehm; Tina Bolvig; Orla Miller Larsson; Arne Schousboe; Povl Krogsgaard-Larsen

Selective Inhibitors of Glial GABA Uptake: Synthesis, Absolute Stereochemistry, and Pharmacology of the Enantiomers of 3-Hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazole (exo-THPO) and Analogues

Erik Falch, Bente Frølund, Perregaard, Connie Sanchez, Birgitte Søkilde, Anders Buur, Anette Hansen, Karla Andrea Frydenvang, Lotte Brehm, Tina Bolvig, Orla Miller Larsson, Arne Schousboe, Povl Krogsgaard-Larsen

Research output: Contribution to journal › Journal article › Research › peer-review

51 Citations (Scopus)

Original language	English
Journal	Journal of Medicinal Chemistry
Volume	42
Pages (from-to)	5402–5414
ISSN	0022-2623
Publication status	Published - 1999

Cite this

Falch, E., Frølund, B., Perregaard, Sanchez, C., Søkilde, B., Buur, A., Hansen, A., Frydenvang, K. A., Brehm, L., Bolvig, T., Larsson, O. M., Schousboe, A., & Krogsgaard-Larsen, P. (1999). Selective Inhibitors of Glial GABA Uptake: Synthesis, Absolute Stereochemistry, and Pharmacology of the Enantiomers of 3-Hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazole (exo-THPO) and Analogues. Journal of Medicinal Chemistry, 42, 5402–5414.

Selective Inhibitors of Glial GABA Uptake: Synthesis, Absolute Stereochemistry, and Pharmacology of the Enantiomers of 3-Hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazole (exo-THPO) and Analogues. / Falch, Erik; Frølund, Bente; Perregaard et al.
In: Journal of Medicinal Chemistry, Vol. 42, 1999, p. 5402–5414.

Research output: Contribution to journal › Journal article › Research › peer-review

Falch, E, Frølund, B, Perregaard, Sanchez, C, Søkilde, B, Buur, A, Hansen, A, Frydenvang, KA, Brehm, L, Bolvig, T, Larsson, OM, Schousboe, A & Krogsgaard-Larsen, P 1999, 'Selective Inhibitors of Glial GABA Uptake: Synthesis, Absolute Stereochemistry, and Pharmacology of the Enantiomers of 3-Hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazole (exo-THPO) and Analogues', Journal of Medicinal Chemistry, vol. 42, pp. 5402–5414.

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title = "Selective Inhibitors of Glial GABA Uptake: Synthesis, Absolute Stereochemistry, and Pharmacology of the Enantiomers of 3-Hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazole (exo-THPO) and Analogues",

author = "Erik Falch and Bente Fr{\o}lund and Perregaard and Connie Sanchez and Birgitte S{\o}kilde and Anders Buur and Anette Hansen and Frydenvang, {Karla Andrea} and Lotte Brehm and Tina Bolvig and Larsson, {Orla Miller} and Arne Schousboe and Povl Krogsgaard-Larsen",

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AU - Falch, Erik

AU - Frølund, Bente

AU - Perregaard, null

AU - Sanchez, Connie

AU - Søkilde, Birgitte

AU - Buur, Anders

AU - Hansen, Anette

AU - Frydenvang, Karla Andrea

AU - Brehm, Lotte

AU - Bolvig, Tina

AU - Larsson, Orla Miller

AU - Schousboe, Arne

AU - Krogsgaard-Larsen, Povl

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JO - Journal of Medicinal Chemistry

JF - Journal of Medicinal Chemistry

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