Abstract
A new tactic for the synthesis and selective functionalization of [1,2,4]triazolo[4,3-a]pyrazines has been developed using an oxidative cyclization as key step. Furthermore, novel strategies for introducing diverse substituents in all positions of the heterocycle were identified.
Original language | English |
---|---|
Journal | SYNLETT: Accounts and Rapid Communications in Chemical Synthesis |
Volume | 26 |
Issue number | 4 |
Pages (from-to) | 519-524 |
Number of pages | 6 |
ISSN | 0936-5214 |
DOIs | |
Publication status | Published - 2015 |
Keywords
- heterocyclic chemistry
- cyclization
- lithiation
- cross-coupling
- PhI(OAc)(2)