Targeting histone lysine demethylases by truncating the histone 3 tail to obtain selective substrate-based inhibitors

Brian Lohse; Anders L Nielsen; Jan B L Kristensen; Charlotte Helgstrand; Paul Andreas Compare Cloos; Lars Olsen; Michael Gajhede; Rasmus Prætorius Clausen; Jesper Langgaard Kristensen

doi:10.1002/anie.201101849

Targeting histone lysine demethylases by truncating the histone 3 tail to obtain selective substrate-based inhibitors

Brian Lohse, Anders L Nielsen, Jan B L Kristensen, Charlotte Helgstrand, Paul Andreas Compare Cloos, Lars Olsen, Michael Gajhede, Rasmus Prætorius Clausen, Jesper Langgaard Kristensen

Research output: Contribution to journal › Journal article › Research › peer-review

36 Citations (Scopus)

Original language	English
Journal	Angewandte Chemie International Edition
Volume	50
Issue number	39
Pages (from-to)	9100-9103
ISSN	1433-7851
DOIs	https://doi.org/10.1002/anie.201101849
Publication status	Published - 19 Sep 2011

Keywords

Former Faculty of Pharmaceutical Sciences
BRIC

Access to Document

10.1002/anie.201101849

Cite this

Targeting histone lysine demethylases by truncating the histone 3 tail to obtain selective substrate-based inhibitors. / Lohse, Brian; Nielsen, Anders L; Kristensen, Jan B L; Helgstrand, Charlotte; Cloos, Paul Andreas Compare; Olsen, Lars; Gajhede, Michael ; Clausen, Rasmus Prætorius ; Kristensen, Jesper Langgaard.

In: Angewandte Chemie International Edition, Vol. 50, No. 39, 19.09.2011, p. 9100-9103.

Research output: Contribution to journal › Journal article › Research › peer-review

Lohse, Brian ; Nielsen, Anders L ; Kristensen, Jan B L ; Helgstrand, Charlotte ; Cloos, Paul Andreas Compare ; Olsen, Lars ; Gajhede, Michael ; Clausen, Rasmus Prætorius ; Kristensen, Jesper Langgaard. / Targeting histone lysine demethylases by truncating the histone 3 tail to obtain selective substrate-based inhibitors. In: Angewandte Chemie International Edition. 2011 ; Vol. 50, No. 39. pp. 9100-9103.

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